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filingDate 2009-10-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-01-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5b60d2307ec3f2e42537aabc77321c91
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publicationDate 2013-01-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8344160-B2
titleOfInvention Pyrrolone melanin concentrating hormone receptor-1 antagonists
abstract The present application provides compounds, including all stereoisomers, solvates, prodrugs and pharmaceutically acceptable forms thereof according to Formula I n nwherein R 1 ,n n nR 4 , R 5 ,n n nR 3 , R 3a , W, D, R 2a , R 2b and R 2c are defined herein.n n Additionally, the present application provides pharmaceutical compositions containing at least one compound according to Formula I and optionally at least one additional therapeutic agent. Finally, the present application provides methods for treating a patient suffering from an MCHR-1 modulated disease or disorder such as, for example, obesity, diabetes, depression, anxiety or intestinal inflammation, by administration of a therapeutically effective dose of a compound according to Formula I.
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Total number of triples: 4027.