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publicationDate 2012-12-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8324204-B2
titleOfInvention Fused thiophene derivatives as kinase inhibitors
abstract A series of 5,6-dihydro-1-benzothiophen-7(4H)-one derivatives, and analogues thereof, which are substituted in the 2-position by an optionally substituted morpholin-4-yl moiety, being selective inhibitors of PI3 kinase enzymes, are accordingly of benefit in medicine, for example in the treatment of inflammatory, autoimmune, cardiovascular, neurodegenerative, metabolic, oncological, nociceptive or ophthalmic conditions.
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Total number of triples: 4005.