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grantDate 2012-10-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2012-10-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8278465-B2
titleOfInvention Coumarin derivative having antitumor activity
abstract The present invention provides a compound represented by general formula (1) below or a pharmaceutically acceptable salt thereof: n nwherein: X is selected from heteroaryl etc., Y 1 and Y 2 are selected from β€”N═ etc., Y 3 and Y 4 are selected from β€”CH═ etc., A is selected from sulfamide etc., R 1 is selected from hydrogen etc., and R 2 is selected from C 1-6 alkyl etc. The compound or salt has sufficiently high antitumor activity, and is useful in the treatment of cell proliferative disorders, particularly cancers. The present invention also provides a pharmaceutical composition containing the compound or salt as an active ingredient.
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Total number of triples: 3988.