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filingDate 2008-03-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2012-08-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8247403-B2
titleOfInvention Benzoxazepine derivatives and use thereof
abstract Compounds represented by the general formula (I): n nwherein each symbol is as defined in the description [with the proviso that 9-chloro-7-(1,1-dimethylethyl)-2,3,4,5-tetrahydro-1,4-benz-oxazepine and N-[[(5S)-2-oxo-3-(2,3,4,5-tetrahydro-1,4-benz-oxazepin-7-yl)-5-oxazolidinyl]methyl]acetamide are excluded], salts of the same, and prodrugs thereof have selective activation effect on serotonin 5-HT 2C receptor and are useful as preventive and therapeutic agents for lower urinary tract diseases, obesity, and/or pelvic organ prolapse.
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Total number of triples: 3277.