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filingDate 2008-04-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2012-05-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2d84b5b67cb5771aab492e596983050f
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publicationDate 2012-05-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8183236-B2
titleOfInvention Compounds with HIV-1 integrase inhibitory activity and use thereof as anti-HIV/AIDS therapeutics
abstract Pharmacophore models to be used in drug design and discovery are provided. An in silico protocol and in vitro assays are presented. Compounds and their pharmaceutically acceptable salts with HIV-1 integrase inhibitory and anti-HIV activity and use thereof in the treatment of HIV/AIDS and related infections either alone or in combination with all the known antiretroviral therapeutics are described.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2013267559-A1
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priorityDate 2007-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57646588
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID327665334
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID123507215
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232417052
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID244
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57646595
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232417051
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID324873120
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57646594
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453049563
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232417049
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449662438
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID324269256
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57646593
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID232417065
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID324871500
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54719422
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449142818
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID324264572

Total number of triples: 2203.