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filingDate 2009-08-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2011-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_17379e06e13dd5425a23db7b9d0c7c30
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_95d051e3c76c04420842ece54c80cfec
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publicationDate 2011-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8063098-B2
titleOfInvention GlyT1 receptor antagonists
abstract The present invention relates to a compound of formula I n nwhereinn R 1 , R 2 , X, Ar 1 and Ar 2 are as defined herein and to pharmaceutically acceptable acid addition salts, to a racemic mixtures, or to their corresponding enantiomers and/or optical isomers thereof. Compounds of the invention are good inhibitors of the glycine transporter 1 (GlyT-1), and have a good selectivity to glycine transporter 2 (GlyT-2) inhibitors.
priorityDate 2008-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 850.