http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-8053457-B2

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grantDate 2011-11-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2011-11-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8053457-B2
titleOfInvention 3-imidazolyl-indoles for the treatment of proliferative diseases
abstract The invention relates to 3-heterocyclyl indolyl compounds of formula I capable of inhibiting the interaction between p53, or variants thereof, and MDM2 and/or MDM4, or variants thereof, respectively: n nwhereinn n R 1 , R 2 , R 3 , R 4 , R A , Y and Y are as defined in the specification. Due to their activity, the compounds are useful in the treatment of various disorders and diseases mediated by the activity of MDM2 and/or MDM4, or variants thereof, such as inflammatory or proliferative diseases or in the protection of cells.
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Total number of triples: 5442.