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publicationDate 2011-10-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-8039472-B2
titleOfInvention Pyrazine-2-carboxamide derivatives to treat diseases mediated by blockade of the epithelial sodium channel
abstract A compound of Formula I n nin free or salt or solvate form, where R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , R 9 , R 10 and R 11 have the meanings as indicated in the specification, is useful for treating diseases which respond to the blockade of the epithelial sodium channel. Pharmaceutical compositions that contain the compounds and processes for preparing the compounds are also described.
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Total number of triples: 3276.