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filingDate 2008-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2011-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7989663-B2
titleOfInvention Compounds and methods of use thereof for assaying lysophospholipase D activity
abstract Fluorogenic lysophosphatidic acid derivatives which can be used as substrates in a continuous, fluorogenic assay that can be performed in microtiter plates. The assays permit measuring LysoPLD activity levels in normal events such as pregnancy or disease states such as cancer. In addition, the present invention can be adopted to high throughout screening (HTS) for identification of potential inhibitors of lysoPLD activity.
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