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filingDate 2005-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2011-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5da64e500b7371a574d897d938309e1f
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publicationDate 2011-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7989624-B2
titleOfInvention Aryl spirolactam CGRP receptor antagonists
abstract The present invention is directed to compounds of Formula (I): where variables A 1 , A 2 , B, J, K, m, n, R 4 , R 5a , R 5b , R 5c and X are as defined herein useful as antagonists of CGRP receptors and useful in the treatment or prevention of diseases in which the CGRP is involved, such as headache, migraine and cluster headache. The invention is also directed to pharmaceutical compositions comprising these compounds and the use of these compounds and compositions in the prevention or treatment of such diseases in which CGRP is involved.
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type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395832
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31101
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128093762
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395726
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24699
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226608790
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12832002
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP97490
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395701
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70934
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226406094
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502484
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419529376
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129349967
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73909
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129313279
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID136100470
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420327887
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5284627
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129347866
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395769
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ76L34
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8119
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID175540
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3059003
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3696
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID161926999
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ76L33
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5816
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419580652
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127658618
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426726972
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129471329
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419581439
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11710798
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11698160
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07660
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504599
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID244466987
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419484695
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128243637
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128133330
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128256022
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395920
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419479746
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226515861
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128133149
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226398848
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID244568790
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395919
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10351092
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226515860
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128253731
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226405997
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID127397498
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14017
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226395921
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504530
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11535
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ57692
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87085720
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WQ35
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WQ34
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID129707927
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08678
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128115633
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID128706830
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID322621738
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226485509

Total number of triples: 1959.