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filingDate 2005-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2011-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6de7bccf70f9069e09abb39663bdaad8
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1f878b344ba1cd42835b5df008b0a4da
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publicationDate 2011-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7960386-B2
titleOfInvention Pyridin-2-one compounds and their use as modulators of the dopamine D3 receptor
abstract The invention relates to pyridin-2-one compounds of general formula (I) n nin whichn A represents a 4- to 6-membered hydrocarbon chain that can have 1 or 2 methyl groups as substituents, wherein 1 or 2 carbon atoms can be replaced by oxygen, a carbonyl group or sulfur, and the hydrocarbon chain can have a double bond or a triple bond; R 1 , R 2 , R 3 and R 4 have the meanings as cited in the claims and in the description. nn The invention also relates to the tautomers of compounds I and the physiologically acceptable salts of the compounds I and their tautomers. n The invention also relates to the use of these compounds for treating diseases that respond to the influence of dopamine D 3 receptor antagonists or agonists.
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Total number of triples: 578.