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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_568dd2c34f318316cc8b3bb7267ac4ac
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publicationDate 2011-03-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7906645-B2
titleOfInvention Heterocyclic compounds as ccr2b antagonists
abstract Compounds of formula (I) Q-L-W—C(═X)—Z—P wherein Q is an amine of the formula —N(R1)(R2); L is an alkyl or heterocyclyl-alkyl linker; W is a 6- or 7-membered aliphatic ring comprising ring atoms Y1 and Y2 which are linked to groups L and C(X) respectively and Y1 and Y2 are independently selected from N and C; X is O, N, N—CN or S; Z is NR3; P is an optionally substituted monocyclic or bicyclic aryl or heteroaryl group; and pharmaceutically acceptable salts or solvates thereof, are useful in the treatment of C-C chemokine mediated conditions.
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Total number of triples: 5015.