http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-7869958-B2

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filingDate 2005-08-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2011-01-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2011-01-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7869958-B2
titleOfInvention Structure-based modulators of B1 G-protein coupled receptors
abstract The present invention relates to a method for identifying modulators of B1 G-protein coupled receptors. The present invention also relates to a method for identifying an antagonist or agonist of the corticotropin-releasing factor receptor 2 (CRFR2). The present invention also relates to a method for improving antagonists or agonists of CRFR2. The present invention also relates to the three-dimensional structure of CRFR2 as representative of the B1 GPCR subfamily and its use as a basis for rational drug design of antagonist or agonists of B1 GPCRs.
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