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publicationDate 2010-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7786119-B2
titleOfInvention Drug conjugates of ion channel modulating compounds
abstract This invention is directed to drug conjugates of certain ion channel modulating compounds having the following formula: n nwherein A, X, R 1 , R 2 , R 3 , R 4 , R 5 , LB, L and DM are defined herein, including isolated enantiomeric and diastereomeric isomers thereof, and mixtures thereof. Pharmaceutical compositions and methods of use are also disclosed.
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Total number of triples: 2067.