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publicationDate 2010-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7785564-B2
titleOfInvention Design and synthesis of renal dipeptidase inhibitors
abstract Aminophosphinic acid derivatives were synthesized as potential inhibitors of renal dipeptidase, an enzyme overexpressed in benign and malignant colon tumors. Several compounds showed potent enzyme-inhibitory activity. These compounds can be used therapeutically and diagnostically for treatment and detection of tumors.
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