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publicationDate 2010-06-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7737145-B2
titleOfInvention Diamine derivatives as inhibitors of leukotriene A4 hydrolase
abstract This invention is directed to compounds of formula (I): n nwhere r, q, R, R 2 , R 3 , R 4 , R 5a , R 5b , R 5c , R 6a , R 6b , R 6c , R 7 , R 8 , and R 9 are described herein, as single stereoisomers or as mixtures of stereoisomers, or pharmaceutically acceptable salts, solvates, clathrates, polymorphs, ammonium ions, N-oxides or prodrugs thereof; which are leukotriene A 4 hydrolase inhibitors and therefore useful in treating inflammatory disorders. Pharmaceutical compositions comprising the compounds of the invention and methods of preparing the compounds of the invention are also disclosed.
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Total number of triples: 2122.