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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1e8f5efcedf1fb615e6779c63134cfc3
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publicationDate 2010-05-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7718653-B2
titleOfInvention Pyrimidine derivatives for inhibiting Eph receptors
abstract A compound of formula (I) n nwhere one of A 1 , A 2 or A 3 is N, and the others are independently selected from CH or N; ring B is a fused 5 or 6-membered carbocyclic or heterocyclic ring which is optionally substituted as defined in the specification, and R 1 , R 2 , R 3 , R 4 , and n are as defined in the specification.n n The compounds are inhibitors of EphB4 or EphA2 and therefore may be useful in pharmaceutical compositions for the treatment of conditions such as cancer.
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8DZM3
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Total number of triples: 1385.