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filingDate 2007-04-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2009-09-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7ddb44ba514100de7c721be69bb47dc3
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5bc3f1deae0c83258c93ca7208a24bf5
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publicationDate 2009-09-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7595317-B2
titleOfInvention Barbituric acid derivatives as inhibitors of TNF-α converting enzyme (TACE) and/or matrix metalloproteinases
abstract The present application describes novel barbituric acid derivatives of formula I: n nor pharmaceutically acceptable salt or prodrug forms thereof, wherein A, B, L, R 1 , R 2 , R 3 , R 4 , R 5 , n, W, U, X, Y, Z, U a , X a , Y a , and Z a are defined in the present specification, which are useful as TNF-α converting enzyme (TACE) and matrix metalloproteinases (MMP) inhibitors.
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priorityDate 2001-12-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 2178.