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filingDate 2008-01-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2009-09-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_52aa051f9a28ade8db464ae5cdbc8648
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publicationDate 2009-09-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7582633-B2
titleOfInvention Azacycloalkane derivatives as inhibitors of stearoyl-coenzyme a delta-9 desaturase
abstract Azacycloalkane derivatives of structural formula I are selective inhibitors of stearoyl-coenzyme A delta-9 desaturase (SCD1) relative to other known stearoyl-coenzyme A desaturases. The compounds of the present invention are useful for the prevention and treatment of conditions related to abnormal lipid synthesis and metabolism, including cardiovascular disease, such as atherosclerosis; obesity; diabetes; neurological disease; metabolic syndrome; insulin resistance; and liver steatosis.
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Total number of triples: 1842.