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filingDate 2007-10-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2009-03-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_052d8143c2232f91013f369bf0d2ab06
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9c896a7e1ccb8877454782d7298ef686
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publicationDate 2009-03-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7501408-B2
titleOfInvention Inhibitors of cathepsin S
abstract The present invention provides compounds, compositions and methods for the selective inhibition of cathepsin S. In a preferred aspect, cathepsin S is selectively inhibited in the presence of at least one other cathepsin isozyme. The present invention also provides methods for treating a disease state in a subject by selectively inhibiting cathepsin S. More particularly, the present invention provides compounds having Formula (I): n n n n n n n n n n n n wherein Q is thiomorpholinyl; and n A, R 5 , R 6 , R 7 , R 8 , R 9 and Ar are substituents.
priorityDate 2003-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226403335
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID142330299
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID242664006
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GLE3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13860
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID228297799
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11478637
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414440311
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID242663932
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226403696
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID142312970
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID245214775
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11387187
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID245119851

Total number of triples: 2196.