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filingDate 2003-08-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2008-04-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2b27b67708fd86e09f488636bf53c711
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c2cd65b455f9f8839aa037037aee3272
publicationDate 2008-04-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7354940-B2
titleOfInvention 2,5-dioxoimidazolidin-4-yl acetamines and analogues as inhibitors of metalloproteinase mmp12
abstract The invention provides compounds of formula (I) in which L, X, Y, Z 1 , Z 2 , R 1 , R 2 , R 3 and G 2 have the meanings defined in the specification; processes for their preparation; pharmaceutical compositions containing them; a process for preparing the pharmaceutical compositions; and their use in therapy. The compounds of the invention are inhibitors of metalloproteinase MMP12 and are among other things useful for the treatment of obstructive airways diseases, such as asthma and chronic obstructive pulmonary disease (COPD).
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Total number of triples: 1516.