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filingDate 2002-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2007-12-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bfbce79dd143cd908cdf73237139ca49
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publicationDate 2007-12-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7312360-B2
titleOfInvention Substituted hydroxyethylamines
abstract Disclosed are compounds of the formula n nand the pharmaceutically acceptable salts thereof wherein the variables G, L, A, W, E, R2, R3, R4, R5, R N , and R c are defined herein. These compounds interact with and inhibit the activity of the enzyme beta-secretase. These compounds are therefore useful in treating Alzheimer's disease and other similar diseases. Pharmaceutical compositions and methods of treatment of these diseases are also disclosed.
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Total number of triples: 2303.