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publicationDate 2007-09-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7268158-B2
titleOfInvention 6H-THIENO [2,3-b]pyrrole derivatives as antagonists of gonadotropin releasing hormone (GnRH)
abstract The invention relates to a group of novel thieno-pyrrole compounds of Formula (I): n nwherein: R 1 , R 2 , R 3 , R 4 and R 5 are as defined in the specification, which are useful as gonadotrophin releasing hormone antagonists. The invention also relates to pharmaceutical formulations of said compounds, methods of treatment using said compounds and to processes for the preparation of said compounds.
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Total number of triples: 3914.