http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-7094789-B2

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D217-04
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-44
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D217-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D217-02
filingDate 2003-07-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2006-08-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_297bccb927a9c80f5f13ec979a1266c2
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ded6ab2c726f21620dd01dacb35e9fbc
publicationDate 2006-08-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7094789-B2
titleOfInvention 5-substituted isoquinoline derivatives
abstract A compound represented by the following formula (1) or a salt thereof: n nwherein R 1 represents hydrogen atom, a halogen atom and the like; R 2 represents hydrogen atom, a halogen atom, a C 1-6 alkyl group and the like; and R 3 represents —O—X—C(A 1 )(A 11 )-C(A 2 )(A 21 )-N(A 31 )(A 3 ) (X represents propylene group etc., A 11 and A 21 represent hydrogen atom, or a C 1-6 alkyl group, A 31 represents a C 1-6 alkyl group substituted with hydroxyl group, or hydrogen atom, and A 1 , A 2 , and A 3 represent hydrogen atom, a C 1-6 alkyl group and the like) and the like, which has an inhibitory activity on the phosphorylation of myosin regulatory light chain, and is useful for treatment of diseases relating to contraction of various cells and the like.
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Total number of triples: 3093.