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publicationDate 2006-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-7033773-B1
titleOfInvention Screening assays for G protein coupled receptor agonists and antagonists
abstract Parathyroid hormone (PTH) and its closely related peptide, PTHrP, share the same receptor, PTHR. LLC-PK1 cells are porcine renal epithelial cells which do not normally express PTHR. The present-invention provides stably transfected LLC-PK1 cells which express human PTHR. Also provided are methods for determining whether a compound of interest is an agonist or antagonist of a Gs or Gq protein coupled receptor.
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