http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-6992193-B2

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filingDate 2003-06-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2006-01-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8f04749a49b2b826d4e08eff129afea3
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1cb1e90fcefb759e7d00f2e161f54ce4
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publicationDate 2006-01-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6992193-B2
titleOfInvention Sulfonylamino phenylacetamide derivatives and methods of their use
abstract Sulfonylamino phenylacetamide derivatives of the general formula n n nare disclosed. Pharmaceutical compositions containing the compounds and methods for their use are also disclosed. In certain embodiments, the compounds of the invention that, preferably:n (1) bind with high affinity to κ opioid receptors; (2) display good opioid receptor selectivity of κ versus μ and κ versus δ; and (3) do not substantially inhibit cytochrome P450 enzymatic activity, in particular CYP2D6, CYP2C9 and CYP3A4.
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Total number of triples: 3333.