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filingDate 2002-06-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2005-11-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2005-11-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6962931-B2
titleOfInvention Self-emulsifying formulations of cholesteryl ester transfer protein inhibitors
abstract CETP Inhibitors have improved solubility and bioavailability in a lipophilic vehicle comprising a digestible oil, a lipophilic solvent, or a surfactant. Preferred such compositions are self-emulsifying or self-microemulsifying, and comprisen 1. a CETP inhibitor; 2. a cosolvent; 3. a surfactant having an HLB of 1 to 8; 4. a surfactant having an HLB of over 8 to 20; and 5. optionally, a digestible oil.
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Total number of triples: 2008.