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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K51-0476
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F13-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K51-04
filingDate 2002-05-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2005-05-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5024dd6eb16808074e52b3b1df7d0173
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_59eef5afe16a88b89b4092a77e89b240
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8a4f1a24fd4c8e940a017549b1bac32d
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publicationDate 2005-05-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6890513-B2
titleOfInvention Metal-carborane complexes for radioimaging and radiotherapy and methods for their preparation
abstract The present invention relates to a new method for the preparation of radiopharmaceuticals based on technetium and rhenium. The method involves the reaction of a salt of the formula [M(CO) 3 (X m ) 3 ] (1+3m) , wherein M is selected from a radioisotope of rhenium, technetium and any other radioisotope that binds in a similar fashion, X is any suitable ligand and m is the formal charge for ligand X, with a nido-dicarbollide dianion of the formula [nido-(C 2 B 9 H 11 )] 2− and functional derivatives thereof. The method has been shown to be applicable to the preparation of radiopharmaceuticals at the tracer level.
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