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filingDate 2001-09-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2005-01-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c2ec0dfde262283b31fbd6fa4143aa9b
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publicationDate 2005-01-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6838479-B2
titleOfInvention Amidine inhibitors of serine proteases
abstract Inhibitors of serine proteases are provided having formula (I) n n nwherein X, R 1 , R 2 , R 3 , R 4 and R 5 are as defined herein. In particular, the compounds bind to factor VIIa, tissue factor/factor Xa complex, thrombin, trypsin, plasmin and kallikrein and have anticoagulant activity. Pharmaceutical compositions comprising the compounds are useful for inhibiting the formation of veinous and/or arterial thrombi in vivo.
priorityDate 2000-09-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 806.