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publicationNumber US-6559158-B1
titleOfInvention Use of methylnaltrexone and related compounds to treat chronic opioid use side affects
abstract A method of preventing or treating an opioid-induced side effect in a patient who has been chronically taking opioids, the method comprising administering a quaternary derivative of noroxymorphone in an amount sufficient to prevent or treat the side effect in the patient, but which amount would be insufficient to treat a patient with the same opioid-induced side effect who had not chronically been administered opioids.
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