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filingDate 1998-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2003-04-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2003-04-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6545022-B1
titleOfInvention 4(3)substituted-4(3)-aminomethyl-(thio)pyran or piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
abstract Novel amines of formulas 1D and 1Eare disclosed and are useful as agents in the treatment of epilepsy, faintness attacks, hypokinesia, cranial disorders, neurodegenerative disorders, depression, anxiety, panic, pain, neuropathological disorders, inflammatory diseases, and gastrointestinal disorders, especially IBS. Processes for the preparation and intermediates useful in the preparation are also disclosed.
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Total number of triples: 703.