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publicationDate 2002-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6495685-B1
titleOfInvention Process for preparing piperazine derivatives
abstract A process for preparing a piperazine derivative represented by the formula (V):comprising reacting 1-methyl-3-phenylpiperazine with 2-chloro-3-cyanopyridine in an aprotic polar organic solvent in the presence of a base and an alkali metal halide. The piperazine derivative and its oxalate are compounds useful as preparation intermediates of mirtazapine.
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