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grantDate 2002-05-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_791ec4791dbc665b6ba1fc53c58c553b
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_01e53eeaf802e843bfe00fae524cfd41
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publicationDate 2002-05-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6387885-B1
titleOfInvention 3′,3′-N-bis-desmethyl-3′-N-cycloalkyl erythromycin derivatives as LHRH antagonists
abstract Disclosed are 3',3'-N-bis-desmethyl-3'-N-cycloalkyl-6-O-methyl-11-deoxy-11,12-cyclic carbamate erythromycin A derivatives which are antagonists of lutenizing hormone-releasing hormone (LHRH). Also disclosed are pharmaceutical compositions comprising the compounds, to methods of using the compounds and to the process of making the same.
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Total number of triples: 428.