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publicationDate 2002-04-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6372736-B1
titleOfInvention Heterocyclic compounds as inhibitors of rotamase enzymes
abstract Compounds of the formula (I):wherein A, Y, R, X, R1, R2, R3 and R4 are as defined above are inhibitors of rotamase enzymes in particular FKBP-12 and FKBP-52. The compounds therefore moderate neuronal regeneration and outgrowth and can be used for treating neurological disorders arising from neurodegenerative diseases or other disorders involving nerve damage.
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Total number of triples: 1157.