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filingDate 1998-06-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2002-04-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6372205-B1
titleOfInvention Pharmaceutical compositions containing antibody-enzyme conjugates in combination with prodrugs
abstract Prodrugs which can be activated by enzymes, are formulated for sequential administration, with enzyme conjugates. Either or each component comprises a polymeric carrier which allows it to be directed preferentially to the target tissue. A new polymer-prodrug conjugate is cleavable by cathepsin-B or othe invention is of particular utility for targeting solid tumours.
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