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filingDate 1999-06-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2002-03-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b3d9576fb346e232c7535c87ec74aabb
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publicationDate 2002-03-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-6358985-B1
titleOfInvention Inhibitors of prenyl-protein transferase
abstract The present invention is directed to peptidomimetic macrocyclic compounds which inhibit prenyl-protein transferase and the prenylation of the oncogene protein Ras. The invention is further directed to chemotherapeutic compositions containing the compounds of this invention and methods for inhibiting prenyl-protein transferase and the prenylation of the oncogene protein Ras.
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Total number of triples: 1798.