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publicationDate 1999-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5972898-A
titleOfInvention 3',3-N-bis-substituted macrolide LHRH antagonists
abstract Disclosed are 3',3'-N-bisdesmethyl-3',3'-N-bis-substituted-6-O-methyl-11-deoxy-11,12 -cyclic carbamate erythromycin A derivatives which are antagonists of lutenizing hormone-releasing hormone (LHRH). Also disclosed are pharmaceutical compositions comprising the compounds, to methods of using the compounds and to the process of making the same.
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Total number of triples: 451.