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filingDate 1994-07-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 1997-06-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fca5f3ca61f680f7a586ae2af688685b
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8ed9dbccda69f61006f4ba09b4a787fa
publicationDate 1997-06-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5641762-A
titleOfInvention Bone targeted inhibitors of carbonic anhydrase
abstract The present invention relates to novel compounds useful for the treatment and prophylaxis of degenerative bone disorders and to the preparation thereof. These compounds are particularly characterized by two active moieties, the first of which possesses "bone-seeking" affinity and the second which is an inhibition of the enzyme carbonic anhydrase and/or an inhibitor of bone resorption. The novel compounds of this invention can be administered as pharmaceutically acceptable compositions and in convenient dosage unit form in a method for the treatment and prophylaxis of degenerative bone disorders.
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