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publicationDate 1997-04-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5622947-A
titleOfInvention Benzoheterocyclic compounds and vasopressin antagonist and oxytocin antagonist compositions containing a benzoheterocyclic compound
abstract PCT No. PCT/JP93/01483 Sec. 371 Date May 25, 1994 Sec. 102(e) Date May 25, 1994 PCT Filed Oct. 15, 1993 PCT Pub. No. WO94/08582 PCT Pub. Date Apr. 28, 1994An object of the present invention is to provide a vasopressin antagonist and oxytocin antagonist. The vasopressing antagonist and oxytocin antagonist according to the present invention contain, as the active ingredient, a benzoheterocyclic compound represented by the general formula (1): <IMAGE> (wherein R1, R2, R3, R4, R5 and the carbon-carbon bond between 4- and 5-positions in the benzoazepine skeleton are the same as defined in claims 1, 2 and 3.) or salt thereof.
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Total number of triples: 3272.