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filingDate 1993-08-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c4cbb0fe7d20819895fe2765c1881d87
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publicationDate 1996-03-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5498609-A
titleOfInvention Benzoazepinyl compounds as oxytocin and vasopressin antagonists
abstract PCT No. PCT/JP93/01082 Sec. 371 Date Apr. 20, 1994 Sec. 102(e) Date Apr. 20, 1994 PCT Filed Aug. 3, 1993 PCT Pub. No. WO94/04525 PCT Pub. Date Mar. 3, 1994.Novel benzoheterocyclic compound of the formula (1): <IMAGE> (1) and pharmaceutically acceptable salts thereof, which show excellent anti-vasopressin activity and oxytocin antagonistic activity, and are useful as a vasopressin antagonist or oxytocin antagonist.
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Total number of triples: 1341.