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publicationDate 1992-04-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5102883-A
titleOfInvention Pyrimidine biosynthesis inhibitors useful as immunosuppressive agents
abstract The pyrimidine biosynthesis inhibitors dichloroallyl lawsone, N-(phosphonoacetyl)-L-aspartic acid (PALA), pyrazofurin, and derivatives thereof, are useful as immunomodulatory and anti-inflammatory agents. Pharmaceutical formulations containing these compounds are useful for the treatment of autoimmune diseases, chronic inflammatory diseases, and of organ transplantation rejections.
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