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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_62a60a478af1aea7383b8d34d840de19
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publicationDate 1992-01-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-5081232-A
titleOfInvention Complexes of tc99m radiopharmaceuticals
abstract Complexes useful as radiopharmaceuticals contain the <99m>Tc-NO moiety and a ligand which confers biological target-seeking properties on the complex. Preferred are mono-cationic complexes, particularly having the formula [<99m>Tc(NO)L2X]<+> where X is halide or pseudohalide and L is a bidentate ligand for Technetium, which have interesting properties for use as heart visualising agents. Examples of ligands include di-(dialkyl and diphenyl)-phosphinoethanes and o-phenylenebisdimethylarsine. The complexes may be made by reacting generator eluate pertechnetate with a hydroxylamine salt and with the ligands, preferably in a single step by providing a reaction mixture containing the three reagents optionally in the presence of a reducing agent.
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