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publicationNumber US-4922007-A
titleOfInvention Process for preparing 4-amino-1-hydroxybutylidene-1,1-bisphosphonic acid or salts thereof
abstract A process for the preparation of 4-amino-1-hydroxybutylidene-1,1-bisphosphonic acid or salts thereof which comprises: (a) reacting 4-aminobutyric acid with a mixture of phosphorous acid and PCl3 in the presence of methanesulfonic acid; and (b) recovering said 4-amino-1-hydroxybutylidene1,1-bisphosphonic acid or salts thereof. e
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