http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-4767744-A
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_56666880a5e2b7703e98a4f9b2d9daf6 |
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-00 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D333-48 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D333-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D333-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D335-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K5-06078 |
| classificationIPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K38-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D335-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K5-065 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D333-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D333-48 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D333-20 |
| filingDate | 1987-02-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 1988-08-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5900336f8ce4d5ca0d1f86933968f120 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a53c4d9b2e2d95911ca04621d0fbf792 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_96ce0e7724f3728353375181d60af506 |
| publicationDate | 1988-08-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | US-4767744-A |
| titleOfInvention | Substituted tyrosyl methionyl dipeptide amides |
| abstract | This invention relates to novel substituted tyrosyl alanine dipeptide amides of the formula: ##STR1## and the pharmaceutically acceptable addition salts thereof, wherein R 1 is --OH, --OCH 3 or lower alkoxy of 1-6 carbon atoms; wherein R 2 and R 3 may be the same or different and represent straight or branched chain lower alkyl of 1-6 carbon atoms; wherein R 4 , R 5 R 9 may be the same or different and represent hydrogen or straight or branched chain lower alkyl having 1-6 carbon atoms; wherein R 6 represents hydrogen, or straight or branched chain lower alkyl of 1-6 carbon atoms, or R 6 may act together with N 6 , C w and either R 7 R 8 to form a cycloamine of the formula: ##STR2## such that between R 7 and R 8 , when one acts to form said cycloamine, the other is hydrogen, or straight or branched chain lower alkyl of 1-6 carbon atoms; wherein when neither R 7 nor R 8 is acting to form said cycloamine, R 7 R 8 act together with C w to form a cycloalkyl of the formula: ##STR3## where n=3, 4, 5; wherein C w represents an asymmetric carbon atom when R 7 and R 8 are not the same and may be racemic or have the D or L configuration; and wherein C v represents an asymmetric carbon atom that may be racemic or that may hve the D or L configuration. n These compounds are useful because they possess analgesic activity in mammals. |
| isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-4933325-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-9640118-A1 |
| priorityDate | 1986-07-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 168.