http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-4000122-A
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_a717ea5b2ac78ac329ab3a9659d834d2 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C243-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-40 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-40 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K5-04 |
| filingDate | 1975-04-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 1976-12-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1eb78ed2e05baa91721eacef75d9b167 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_57c67a84b4cd0f4e47d6fd84bfe42eca http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_82b934a1fc1cbc22bd9666de09203b16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b072016dc4cbaf05536527fb40e61af5 |
| publicationDate | 1976-12-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | US-4000122-A |
| titleOfInvention | Novel hydrazinocarboxamide derivatives and preparation thereof |
| abstract | α-Hydrazinocarboxamide and α-(α'-acylhydrazino)-carboxamide derivatives of formula I ##STR1## in which R 1 and R 2 each are lower alkyl or R 1 and R 2 together with the nitrogen atom to which they are joined form a piperidino or morpholino radical; R 3 is hydrogen, lower alkanoyl, benzoyl, p-nitrobenzoyl, p-aminobenzoyl, p-chlorobenzoyl, isocyanoacetyl, or protected amino acyl radicals, for example, N-formylglycyl or ##STR2## (N-carbobenzoxyglycylglycyl); R 4 is lower alkyl, CHR 7 COOR 8 or CH 2 CH 2 COOR 8 wherein R 7 is hydrogen or phenyl and R 8 is hydrogen or lower alkyl; R 5 is hydrogen or lower alkyl; or R 4 and R 5 together with the carbon atom to which they are joined form a cyclohexylidene radical; and R 6 is a cyclohexyl or CHR 9 COY wherein R 9 is hydrogen or benzyl and Y is hydroxyl, lower alkoxy or amine, with the provisos that when Y is hydroxyl then R 8 is hydrogen, that when Y is lower alkoxy than R 8 is lower alkyl and that when Y is amino R 4 is lower alkyl, are disclosed herein along with the related α-hydrazino-carboxamide and α-(α'-acylhydrazino)carboxamide compounds of formula III ##STR3## in which R 1 , R 2 , R 3 , R 5 and R 7 are as defind above and Y is lower alkoxy. These compounds possess antibacterial activity. Methods for their preparation and use are disclosed also. |
| isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-114515606-A |
| priorityDate | 1973-02-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 379.