http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2022281970-A1

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filingDate 2019-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8c3530ba0bd13f6173bedbac32aaf31d
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publicationDate 2022-09-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2022281970-A1
titleOfInvention Pharmaceutical Combinations
abstract The present invention relates to the combination of the HDM2-p53 interaction inhibitor drug (S)-5-(5-Chloro-1-methyl-2-oxo-1,2-dihydro-pyridin-3-yl)-6-(4-chloro-phenyl)-2-(2,4-dimethoxy-pyrimidin-5-yl)-1-isopropyl-5,6-dihydro-1H-pyrrolo[3,4-d]imidazol-4-one [HDM201] and an anti-TIM-3 antibody molecule as TIM-3 inhibitor. The present invention further relates to the use of said combination in the treatment of cancer, in particular hematological tumors. The present invention further relates to dose and dosing regimen related to this combination cancer treatment.
priorityDate 2018-12-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95KP3
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59750
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID83817
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8D4H3
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID737808
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1C6T8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3FEW8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8MKH2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95253
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07750
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04058
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ48727
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3458
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5MBA8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81800
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7KGA5
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397276
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403869
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ04745
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81650
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25712
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6D736
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ07885
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503036
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM5
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403693
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81156
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281248
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP46652
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422454219
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24978538
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4U313
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ03WL0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16168
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID30323
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP46649
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID42890
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7LZG1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4U0U2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCAAA68151
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28028
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6LL68
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID478720255
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22023293
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID394198
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5PXD0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9R0J8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280795
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID405790
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP24131
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2VHN8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422987404
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID449517
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID114549
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16992
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP02701
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO77762
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM3
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9844
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25670
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO77620
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419556509
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID100658
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281237
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8627545
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID456893
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419555131
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403416
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403801
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID109644000
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP56161
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5F5U6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29126
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9840
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ86GC8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0TKT1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6253
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73909
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48982
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48981
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7CIZ3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23989
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9838
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP16278
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID80380
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48980
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22303
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5281426
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID742141
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8AKB8
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID30538
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9MQ82
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCJ9P745
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCJ9NSP1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP36196
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19114
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ86GC9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13308
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ25BC3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10154
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12043
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ865Y1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID574282
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP42202
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID656655
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ865Y0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397926
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID314856
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419529509
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281542
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8X685
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19147
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ867X3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426079013
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396200
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16183
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68291
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21836
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60533
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8AB22
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ47077
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396282
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11423
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP61125

Total number of triples: 464.