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filingDate 2022-01-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2022-07-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2022220078-A1
titleOfInvention Small molecule inhibitors of lactate dehydrogenase and methods of use thereof
abstract Provided is a compound of formula (I)in which Ar1, R1, U, V, W, X, and p are as described herein. Also provided are methods of using a compound of formula (I), including a method of treating cancer, a method of treating a patient with cancer cells resistant to an anti-cancer agent, and a method of inhibiting lactate dehydrogenase A (LDHA) and/or lactate dehydrogenase B (LDHB) activity in a cell.
priorityDate 2014-12-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457593
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163659
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457592
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396559
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318964
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5746
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457595
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396558
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318959
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457594
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1D2L9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318958
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16832
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457589
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318961
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16828
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457588
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318960
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457591
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318955
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457590
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318954
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70146
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457585
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2SJJ1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162318312
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318957
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162323542
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457584
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457587
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162323551
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162325556
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457586
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318950
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457581
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5743
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457580
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54676228
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457583
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318947
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158026224
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457582
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457577
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318949
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5EV80
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457576
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396819
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139318948
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457579
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1RDV1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457578
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162325526
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ21697
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457637
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396820
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457636
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457639
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID157833257
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457638
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457633
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VR40
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457632
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162331947
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226396787
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID226427184
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457635
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID80641327
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457634
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID158285160
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4336216
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457866
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457629
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO67161
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457628
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5790
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457631
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457630
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID65628
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID228793599
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457625
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID148278157
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457624
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162095
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457627
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457626
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27726
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457858
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457621
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457853
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457620
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID162338092
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457623
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121457622
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID244663
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8622873

Total number of triples: 3191.