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filingDate 2021-11-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9dc9a74770365c51f179746676e63bb9
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publicationDate 2022-05-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2022143188-A1
titleOfInvention Formulation for oral delivery of proteins, peptides and small molecules with poor permeability
abstract The present disclosure is directed to a pharmaceutical formulation intended for oral delivery of synthetic or natural poorly permeable molecules or salts/solvates thereof having a therapeutic activity. The pharmaceutical formulation can include a synthetic or natural poorly permeable molecule or salt or solvate thereof in an amount 0.01-10 wt. % of the total weight of the formulation; a lipophilic phase comprising triglycerides of fatty acids in an amount of 50-80 wt. % of the total weight of the formulation; and at least one lipophilic surfactant comprising partial esters of polyol and fatty acids in an amount of about 10-50 wt. % of the total weight of the formulation.
priorityDate 2019-04-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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