http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2022071985-A1

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filingDate 2019-12-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d3e614ca735a113979c3f22f2e651bde
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publicationDate 2022-03-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2022071985-A1
titleOfInvention Quinoline derivatives for use in the treatment or prevention of cancer
abstract A compound of formula (Ib′) or anyone of its metabolites or a pharmaceutically acceptable salt thereof for use for treating and/or preventing cancer and/or dysplasia n n n n n n n n n n wherein R is independently hydrogen, halogen, —CN, hydroxyl, (C 1 -C 3 )fluoroalkyl, (C 1 -C 3 )fluoroalkoxy, (C 3 -C 6 )cycloalkyl, —NO 2 , —NR 1 R 2 , (C 1 -C 4 )alkoxy, phenoxy, —NR 1 —SO 2 —NR 1 R 2 , —NR 1 —SO 2 —R 1 , —NR 1 —C(═O)—R 1 , —NR 1 —C(═O)—NR 1 R 2 , —SO 2 —NR 1 R 2 , —SO 3 H, —O— SO 2 —OR 3 , —O—P(═O)(OR 3 )(OR 4 ), —O—CH 2 —COOR 3 , (C 1 -C 3 )alkyl, said alkyl being optionally mono- or di-substituted by a hydroxyl group, a -A-(CH 2 ) m —B—NRaRb group, or a —(O—CH 2 —CH 2 ) p —O—Ra group. The present disclosure also relates to a compound of formula (IVb′) or a pharmaceutically acceptable salt thereof for use for treating and/or preventing cancer and/or dysplasia.
priorityDate 2018-12-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163781988
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9606
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658892
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2TG13
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420848480
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502374
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Y251
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658893
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2T9B1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118674403
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658890
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ397E7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433754319
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25619
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411675801
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658888
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118674401
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554287
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7FMH4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658889
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5MBA8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3NN77
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6505803
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID49846579
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658887
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2726
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57379345
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15723640
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658884
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413040209
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658885
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5EWS3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408105837
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7FLH4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658882
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8AGR2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25589
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554174
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280822
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658881
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408092222
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO02837
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658878
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47717
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658879
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4EWA3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6918295
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118658876
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4ZVE4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5ETU8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID374569
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2PE78
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6WRB7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411843290
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465179962
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8YSZ5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480599
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID695
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2PE47
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID56069
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67987356
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12229
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480871
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5F9H5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4EUR1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506748
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407287363
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411811319
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4ZU37
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67987354
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6WQU2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67987351
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152743162
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID35199
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID95839
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID888013
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8A8B1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID153274811
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5BAJ8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP60569
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465829075
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ47BM2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4EPB7
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID114781
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152743158
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44631912
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID446541
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4ELA5

Total number of triples: 1646.