http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-2022064161-A1

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filingDate 2020-01-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_686a72e2026f0f3ac9f0773314355152
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publicationDate 2022-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber US-2022064161-A1
titleOfInvention Pyrrolopyridine derivative and use thereof in prevention and treatment of protein kinase-related disease
abstract The present invention relates to a pyrrolopyridine derivative and a pharmaceutical composition comprising the same as an active ingredient for prevention or treatment of a protein kinase-related disease. The pyrrolopyridine derivative has excellent inhibitory activity against various protein kinases including LRRK2, DYRK1, and CLK1 and exhibits an excellent suppressive effect on the growth of triple-negative breast cancer cells. A pharmaceutical composition comprising the same as an active ingredient can be advantageously used for treating or preventing protein kinase-related diseases, inter alia, cancers, degenerative brain diseases, and inflammatory diseases, and specifically for treating triple-negative breast cancer.
priorityDate 2019-01-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1772.